Tegeprotafib
CAS No. : 2407610-46-0
(Synonyms: PTPN2/1-IN-1)
| Size | Price | Stock |
|---|---|---|
| 1mg | $520 | In-stock |
| 5mg | $1160 | In-stock |
| 10mg | $1550 | In-stock |
| 25mg | $2360 | In-stock |
| 50mg | $3080 | In-stock |
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| Cat. No. : | HY-153446 |
| M.Wt: | 326.30 |
| Formula: | C13H11FN2O5S |
| Purity: | >98 % |
| Solubility: | DMSO : 100 mg/mL (ultrasonic) |
Tegeprotafib (PTPN2/1-IN-1) (Compound 124) is an orally active PTPN1 and PTPN2 inhibitor with IC50s of 4.4 nM and 1-10 nM against PTPN2 and PTP1B, respectively[1]. IC50 & Target:IC50: 4.4 nM (PTPN2), 1-10 nM (PTP1B)[1] In Vitro: Tegeprotafib (Compound 124; 5 days) inhibits IFNγ (0.5 ng/mL) induced B16F10 cellular growth with a percent growth inhibition of 60-90% at 33 μM[1]. In Vivo: Tegeprotafib (Compound 124; 300 mg/kg; oral; BID for 21 days) shows antitumor activity in mice[1].
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