OP-1074
CAS No. : 1443752-76-8
| Size | Price | Stock |
|---|---|---|
| 5mg | $850 | In-stock |
| 10mg | $1450 | In-stock |
| 25mg | $2950 | In-stock |
| 50 mg | Get quote | |
| 100 mg | Get quote | |
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| Cat. No. : | HY-125263 |
| M.Wt: | 457.56 |
| Formula: | C29H31NO4 |
| Purity: | >98 % |
| Solubility: | DMSO : 100 mg/mL (ultrasonic) |
OP-1074 is a pure antiestrogen and a selective ER degrader (PA-SERD), shows specific antiestrogenic activity for ERα and ERβ, inhibits 17β-estradiol (E2)-stimulated transcriptional activity with IC50 of 1.6 and 3.2?nM, respectively[1]. In Vitro: OP-1074 (0-100?nM; 24 hours) inhibits ?MCF-7 cells? and CAMA-1 cells proliferation?with IC50 values of 6.3 and 9.2 nM, respectively[1]. OP-1074 (100?nM; 24 hours) destabilizatizes ERα protein expression in MCF-7 and CAMA-1 cells[1].
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