TP-238
CAS No. : 2415263-04-4
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| Cat. No. : | HY-114205 |
| M.Wt: | 458.58 |
| Formula: | C22H30N6O3S |
| Purity: | >98 % |
| Solubility: | 10 mM in DMSO |
TP-238 is a potent and selective dual CECR2/BPTF probe with IC50 values of 30 nM and 350 nM, respectively. TP-238 also inhibits BRD9 with a pIC50 of 5.9 and is less active against other 338 kinases[1][2]. In Vitro: TP-238 has on target biochemical activity of 10-30 nM with CECR2 and 100-350 nM with BPTF. TP-238 displays potency for both CECR2 (pIC50 of 7.5) and BPTF (pIC50 of 6.5) in an Alpha screen assay. Isothermal titration calorimetry (ITC) shows TP-238 with a Kd of 10 nM for CECR2 and 120 nM for BPTF[1][2].
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- TP-238
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- HY-114205
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