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|---|---|---|
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| 500 mg | Get quote | |
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| Cat. No. : | HY-111583 |
| M.Wt: | 383.87 |
| Formula: | C20H22ClN5O |
| Purity: | >98 % |
| Solubility: | 10 mM in DMSO |
RXFP3/4 agonist 1 is an agonist of relaxin family peptide 3/4 receptor (RXFP3/4), with EC50s of 82/2 nM, respectivley. RXFP3/4 agonist 1 increases food intake in rats[1]. IC50 & Target: EC50: 82 nM (RXFP3), 2 nM (RXFP4)[1] In Vitro: RXFP3/4 agonist 1 (Compound 4) inhibits orskolin-stimulated cAMP accumulation in CHO-K1 cells stably overexpressing RXFP3 and RXFP4, with EC50s of 12.8 and 1.6?nM, respectively[1].
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