KDM2A/7A-IN-1
CAS No. : 2169272-46-0
| Size | Price | Stock |
|---|---|---|
| 1mg | $320 | In-stock |
| 5mg | $780 | In-stock |
| 10mg | $1200 | In-stock |
| 25mg | $2400 | In-stock |
| 50mg | $3340 | In-stock |
| 100mg | $4400 | In-stock |
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| 500 mg | Get quote | |
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| Cat. No. : | HY-108706 |
| M.Wt: | 506.68 |
| Formula: | C33H38N4O |
| Purity: | >98 % |
| Solubility: | DMSO : 200 mg/mL (ultrasonic) |
KDM2A/7A-IN-1 is a first-in-class, selective and cell-permeable inhibitor of histone lysine demethylases KDM2A/7A, with an IC50 of 0.16?μM for KDM2A, exhibits 75 fold selevtivity over other JmjC lysine demethylases, and is inactive on methyl transferases, and histone acetyl transferases[1].
IC50 & Target: IC50: 0.16?μM (KDM2A)[1]
In Vitro: KDM2A/7A-IN-1 ((S,S)-6) is a first-in-class, selective and cell-permeable inhibitor of histone lysine demethylases KDM2A/7A, with an IC50 of 0.16?μM for KDM2A, exhibits 75 fold selevtivity over other JmjC lysine demethylases, and is inactive to methyl transferases, and histone acetyl transferases[1].
KDM2A/7A-IN-1 (0.4, 3.1, 6.2 μM) augments cellular H3K36me2 levels in HeLa cells ectopically expressing catalytically active KDM2A[1].
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