PSB-12379 (disodium)
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|---|---|---|
| 100 mg | Get quote | |
| 250 mg | Get quote | |
| 500 mg | Get quote | |
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| Cat. No. : | HY-100747A |
| M.Wt: | 559.31 |
| Formula: | C18H21N5Na2O9P2 |
| Purity: | >98 % |
| Solubility: | 10 mM in DMSO |
PSB-12379 disodium, a nucleotide analogue, is a potent Ecto-5'-Nucleotidase (CD73) inhibitor with Kis of 9.03 nM (rat) and 2.21 nM (human)[1][2]. IC50 & Target:Ki: 9.03 nM (rat), 2.21 nM (human) (Ecto-5’-Nucleotidase)[1]. In Vivo: Metabolism: Only a small percentage (<23%) of PSB-12379 (10g) is metabolized under the applied conditions, while >77% of the compounds are recovered unchanged after a long incubation for 8 h. PSB-12379 (10g) is somewhat less stable, and 56% are metabolized within 8 h. Hydrolytic cleavage of the glycosidic bond, which is a typical phase I reaction of nucleosides and nucleotides, was observed as the main reaction[1].
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Inquiry Information- Product Name:
- PSB-12379 (disodium)
- Cat. No.:
- HY-100747A
- Quantity:
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