2-PCCA
CAS No. : 1984859-71-3
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| Cat. No. : | HY-100013 |
| M.Wt: | 455.63 |
| Formula: | C30H37N3O |
| Purity: | >98 % |
| Solubility: | 10 mM in DMSO |
2-PCCA is a racemic form of the GPR88 receptor agonist, and inhibits GPR88-mediated cAMP production, with an EC50 of 116 nM in HEK293 cells. IC50 & Target:EC50: 116 nM (GPR88 receptor, HEK293 cells)[1] In Vitro:2-PCCA inhibits GPR88-mediated cAMP production through a Gαi-coupled pathway, with an EC50 of 116 nM in HEK293 cells stably expressing the human GPR88 receptor and the GloSensor-22F cAMP construct[2]. In Vivo:2-PCCA (0.1–3.2 mg/kg, intraperitoneal injection) dose-dependently reduces kinetic activity in rats. 2-PCCA (1–3.2 mg/kg, intraperitoneal injection) does not produce a discriminative stimulus effect in rats[1].
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