CH5015765
CAS No. : 959766-47-3
| Size | Price | Stock |
|---|---|---|
| 5mg | $290 | In-stock |
| 10mg | $465 | In-stock |
| 25mg | $930 | In-stock |
| 50mg | $1490 | In-stock |
| 100mg | $2390 | In-stock |
| 200 mg | Get quote | |
| 500 mg | Get quote | |
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| Cat. No. : | HY-111007 |
| M.Wt: | 344.82 |
| Formula: | C16H13ClN4OS |
| Purity: | >98 % |
| Solubility: | DMSO : 50 mg/mL (ultrasonic) |
CH5015765 is an orally available Hsp90 inhibitor bound to the N-terminal ATP binding site, with a dissociation constant of 3.4 nM, CH5015765 exerts antiproliferative activity against human cancer cell lines, with IC50 values of 0.46 μM for HCT116 colorectal cancer cells and 0.57 μM for NCI-N87 gastric cancer cells. CH5015765 can be used for the study of cancer[1][2].
In Vitro:CH5015765 (4 days) exerts in vitro antiproliferative activity against human cancer cell lines, with IC50 values of 0.46 μM for HCT116 colorectal cancer cells and 0.57 μM for NCI-N87 gastric cancer cells[1].
In Vivo:CH5015765 (400 mg/kg, p.o., once daily for 11 consecutive days, Days 11-21) exerts moderate antitumor efficacy in SCID mice bearing human NCI-N87 gastric cancer xenografts[1].
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