TC-E 5005
CAS No. : 959705-64-7
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| Cat. No. : | HY-10568 |
| M.Wt: | 270.33 |
| Formula: | C15H18N4O |
| Purity: | >98 % |
| Solubility: | 10 mM in DMSO |
TC-E 5005 is a potent and selective PDE10A inhibitor with IC50 values of 7.28, 239, 779, 919, 3,100, and 3,700 nM for PDE10A, 2A, 11A, 5A, 7B and 3A, respectively. TC-E 5005 inhibits adrenergic and neurogenic smooth muscle contractions in the human prostate[1].
In Vitro: TC-E 5005 (500 nM) inhibits norepinephrine or phenylephrine and EFS (electric field stimulation)-induced contraction of human prostate strips[1].
TC-E 5005 (500 nM) shows amplification of treprostinil-induced relaxations, which were significant from 0.03 to 30 μM treprostinil[1].
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