Pavinetant
CAS No. : 941690-55-7
(Synonyms: MLE-4901; AZD2624; AZD4901)
| Size | Price | Stock |
|---|---|---|
| 5mg | $220 | In-stock |
| 10mg | $330 | In-stock |
| 50mg | $550 | In-stock |
| 100mg | $810 | In-stock |
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| Cat. No. : | HY-14432 |
| M.Wt: | 459.56 |
| Formula: | C26H25N3O3S |
| Purity: | >98 % |
| Solubility: | DMSO : ≥ 50 mg/mL |
Pavinetant (MLE-4901) is a neurokinin-3 receptor (NK3R) antagonist. IC50 & Target: NK3R[1] In Vitro: Pavinetant (AZD2624) is a potent and selective NK3 receptor antagonist which is developed for the treatment of schizophrenia. Pavinetant exhibits an inhibitory effect on microsomal CYP3A4/5 activities with apparent IC50 values of 7.1 and 19.8 μM for midazolam and testosterone assays, respectively. No time-dependent inactivation of CYP3A4/5 activity by Pavinetant is observed. Pavinetant demonstrates weak to no inhibition of CYP1A2, CYP2B6, CYP2C8, CYP2C9, CYP2C19, and CYP2D6[1].
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