MK-1925
CAS No. : 932705-04-9
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| Cat. No. : | HY-122561 |
| M.Wt: | 362.40 |
| Formula: | C19H21F3N4 |
| Purity: | >98 % |
| Solubility: |
MK-1925 (compound 39) is a ORL1 receptor antagonist with human IC50 values of 8.2 nM and 4.6 nM, as well as oral bioavailability and blood-brain barrier penetration. MK-1925 selectively inhibits the ORL1 receptor and shows no significant activity against other opioid receptors or the hERG potassium channel[1].
In Vitro:MK-1925 (compound 39) is highly selective for ORL1 receptors over human μ, κ, and δ opioid receptors, with ORL1 binding IC50 of 8.2 nM and minimal binding to other opioid receptors (IC50 values ≥9800 nM or >10,000 nM)[1].
MK-1925 has minimal binding affinity for hERG potassium channels, with an IC50 of 9500 nM[1].
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