| Size | Price | Stock |
|---|---|---|
| 5mg | $108 | In-stock |
| 10mg | $156 | In-stock |
| 25mg | $336 | In-stock |
| 50 mg | Get quote | |
| 100 mg | Get quote | |
| We match the lowest price on market. | ||
We offer a substantial discount on larger orders, please inquire via [email protected]
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Inquiry for price and availability only. Please place your order via our email or fax.
| Cat. No. : | HY-P0079 |
| M.Wt: | 745.95 |
| Formula: | C38H63N7O8 |
| Purity: | >98 % |
| Solubility: | H2O : 50 mg/mL (ultrasonic) |
Neuromedin N is a potent modulator of dopamine D2 receptor agonist binding in rat neostriatal membranes. IC50 & Target: Dopamine D2 receptor[1]. In Vitro: Neuromedin N competitively inhibits the binding of neurotensin to rat brain synaptic membranes with a 19-fold lower potency than neurotensin and is rapidly inactivated by brain synaptic peptidases[1]. It competitively inhibits neurotensin binding to rat brain synaptic membranes and has increased potency in the presence of the peptidase inhibitor bestatin[2].
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