CPUY074020
CAS No. : 902279-44-1
| Size | Price | Stock |
|---|---|---|
| 5mg | $190 | In-stock |
| 10mg | $275 | In-stock |
| 25mg | $425 | In-stock |
| 50mg | $600 | In-stock |
| 100mg | $785 | In-stock |
| 200 mg | Get quote | |
| 500 mg | Get quote | |
| We match the lowest price on market. | ||
We offer a substantial discount on larger orders, please inquire via [email protected]
or Fax: (86)21-58955996
Inquiry for price and availability only. Please place your order via our email or fax.
| Cat. No. : | HY-100757 |
| M.Wt: | 416.52 |
| Formula: | C25H28N4O2 |
| Purity: | >98 % |
| Solubility: | 10 mM in DMSO |
CPUY074020 is a potent and oral bioavailable inhibitor of histone methyltransferase G9a, with an IC50 of 2.18 μM. CPUY074020 possesses anti-proliferative activity[1].
IC50 & Target: IC50: 2.18 μM (G9a)[1]
In Vitro: CPUY074020 (2-8μM; 24 hours) induces cell death through apoptosis[1].
CPUY074020 (2.5-10μM ; 48 hours) dose-dependently de-regulates H3K9 trimethylation[1].
In Vivo: CPUY074020 exhibits reasonable PK properties, with an oral bioavailability of 55.5% and a T1/2 value of 4.0 hours at an oral dose of 10 mg/kg[1].
Lorem ipsum dolor sit amet, consectetur adipisicing elit. Autem earum hic iste maiores, nam neque rem suscipit. Adipisci consequatur error exercitationem fugit ipsam optio qui, quibusdam repellendus sed vero! Debitis.
Inquiry Information- Product Name:
- CPUY074020
- Cat. No.:
- HY-100757
- Quantity:
Your information is safe with us.