GSK-5959
CAS No. : 901245-65-6
| Size | Price | Stock |
|---|---|---|
| 5mg | $66 | In-stock |
| 10mg | $110 | In-stock |
| 50mg | $319 | In-stock |
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| 200 mg | Get quote | |
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| Cat. No. : | HY-18665 |
| M.Wt: | 394.47 |
| Formula: | C22H26N4O3 |
| Purity: | >98 % |
| Solubility: | DMSO : 13 mg/mL (ultrasonic;warming) |
GSK-5959 is a potent, selective and cell permeable BRPF1 bromodomain inhibitor with an IC50 of ~ 80 nM[1].
IC50 & Target: IC50: 80 nM (BRPF1)[1].
In Vitro: GSK-5959 (3a) also displays selectivity over the closely related family members, BRPF2 (100-fold) and BRPF3 (>1000-fold)[2].
GSK-5959 (3a) exhibits an EC50 = 0.98 μM) in cellular NanoBRET assay[2].
GSK-5959 has no effect on TRIM24 SUMOylation[3].
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