Deltazinone 1
CAS No. : 894554-89-3
| Size | Price | Stock |
|---|---|---|
| 5mg | $650 | In-stock |
| 10mg | $1050 | In-stock |
| 25mg | $1900 | In-stock |
| 50mg | $3000 | In-stock |
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| 200 mg | Get quote | |
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| Cat. No. : | HY-108436 |
| M.Wt: | 457.57 |
| Formula: | C27H31N5O2 |
| Purity: | >98 % |
| Solubility: | 10 mM in DMSO |
Deltazinone 1, a pyrazolopyridazinone, is a highly selective PDEδ inhibitor with a KD of 8 nM. Deltazinone 1 inhibits the PDEδ-Ras interaction. Deltazinone 1 shows a dose-dependent inhibitory response on proliferation in oncogenic KRas-dependent cell lines[1][2].
In Vitro:Deltazinone 1 (0.375-24 μM; 0-120 h) inhibits cell growth in a dose-dependent manner[1].
Deltazinone 1 (20 μM; 1 h) reduces S6P phosphorylation in the KRas-dependent Panc-Tu-I cells[1].
Deltazinone 1 (10 μM) shows cell death for oncogenic KRas-dependent Panc-Tu-I cells but not for oncogenic KRas-independent PANC-1 cells[1].
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