Size | Price | Stock |
---|---|---|
5mg | $65 | In-stock |
10mg | $110 | In-stock |
25mg | $220 | In-stock |
50mg | $360 | In-stock |
100mg | $580 | In-stock |
200 mg | Get quote | |
500 mg | Get quote | |
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Cat. No. : | HY-100214 |
M.Wt: | 349.41 |
Formula: | C19H15N3O2S |
Purity: | >98 % |
Solubility: | 10 mM in DMSO |
EAI001 is a potent, selective mutant epidermal growth factor receptor (EGFR) allosteric inhibitor with an IC50 value of 24 nM for EGFRL858R/T790M. EAI001 can be used for research of cancer[1][2]. In Vitro: EAI001 (50 μM) binds to EGFR T790M/C797S/V948R that lies deep inside the EGFR towards the ATP binding site and C-helix. EAI001 showed inhibitory activity due to hydrophobic interaction with amino acid Ile759, Leu747, Leu788, Leu777 and Met766[1].
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