EAI001


CAS No. : 892772-75-7

892772-75-7
Price and Availability of CAS No. : 892772-75-7
Size Price Stock
5mg $65 In-stock
10mg $110 In-stock
25mg $220 In-stock
50mg $360 In-stock
100mg $580 In-stock
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Cat. No. : HY-100214
M.Wt: 349.41
Formula: C19H15N3O2S
Purity: >98 %
Solubility: 10 mM in DMSO
Introduction of 892772-75-7 :

EAI001 is a potent, selective mutant epidermal growth factor receptor (EGFR) allosteric inhibitor with an IC50 value of 24 nM for EGFRL858R/T790M. EAI001 can be used for research of cancer[1][2]. In Vitro: EAI001 (50 μM) binds to EGFR T790M/C797S/V948R that lies deep inside the EGFR towards the ATP binding site and C-helix. EAI001 showed inhibitory activity due to hydrophobic interaction with amino acid Ile759, Leu747, Leu788, Leu777 and Met766[1].

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