Efaroxan (hydrochloride)
CAS No. : 89197-00-2
| Size | Price | Stock |
|---|---|---|
| 5mg | $25 | In-stock |
| 10mg | $35 | In-stock |
| 25mg | $70 | In-stock |
| 50mg | $110 | In-stock |
| 100mg | $175 | In-stock |
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| Cat. No. : | HY-B1416A |
| M.Wt: | 252.74 |
| Formula: | C13H17ClN2O |
| Purity: | >98 % |
| Solubility: | DMSO : 50 mg/mL (ultrasonic;warming;heat to 60°C) |
Efaroxan hydrochloride is a potent, selective and orally active α2-adrenoceptor antagonist, with antidiabetic activity. Efaroxan hydrochloride is a selective I1-Imidazoline receptor antagonist. Efaroxan hydrochloride can be used for the research of cardiovascular disease[1][2][3].
IC50 & Target: α2-adrenoceptor, I1-Imidazoline receptor[1][2]
In Vitro: Efaroxan hydrochloride binds to I1-imidazoline and α2-adrenergic receptors in bovine rostral ventrolateral medulla membranes, with Kis of 0.15 nM and 5.6 nM, respectively[1]
In Vivo: Efaroxan hydrochloride increases plasma insulin levels in both conscious fed and fasted rats without greatly affecting plasma glucoselevels[3].
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