CCT129957
CAS No. : 883098-58-6
| Size | Price | Stock |
|---|---|---|
| 5mg | $110 | In-stock |
| 10mg | $165 | In-stock |
| 25mg | $297 | In-stock |
| 50mg | $445 | In-stock |
| 100mg | $668 | In-stock |
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| Cat. No. : | HY-111208 |
| M.Wt: | 309.32 |
| Formula: | C17H15N3O3 |
| Purity: | >98 % |
| Solubility: | DMSO : 100 mg/mL (ultrasonic) |
CCT129957 is an indole derivative and a potent phospholipase C-γ (PLC-γ) inhibitor with an IC50 of ~3 μM and a GC50 of 15 μM. CCT129957 inhibits Ca2+ release in squamous carcinoma cells at ~15 μM[1][2].
IC50 & Target: IC50: ~3 μM (Phospholipase C-γ (PLC-γ))[1]
In Vitro: The phenyl group on the left side sat in a lipophilic pocket formed of various amino acids. The predicted binding mode of CCT129957 displays a robust hydrogen bond pattern as well as a lipophilic contact[1].
CCT129957 inhibits the cell growth of renal UO-31 and the breast T-47D cancer cell lines by ~60-70%[2].
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