Malantide
CAS No. : 86555-35-3
| Size | Price | Stock |
|---|---|---|
| 5mg | $180 | In-stock |
| 10mg | $280 | In-stock |
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| Cat. No. : | HY-P1597 |
| M.Wt: | 1633.89 |
| Formula: | C72H124N22O21 |
| Purity: | >98 % |
| Solubility: | DMSO : 100 mg/mL (ultrasonic) |
Malantide is a synthetic dodecapeptide derived from the site phosphorylated by cAMP-dependent protein kinase (PKA) on the β-subunit of phosphorylase kinase. Malantide is a highly specific substrate for PKA with a Km of 15 μM and shows protein inhibitor (PKI) inhibition >90% substrate phosphorylation in various rat tissue extracts[1]. Malantide is also an efficient substrate for PKC with a Km of 16 μM[2].
IC50 & Target:Km: 15 μM (PKA)[1], 16 μM (PKC)[2], 233 μM (PKG)[1]
In Vitro: The Km values of Malantide are 15 μM and 223 μM for PKA and PKG, respectively. The Vmax values are 23.8 units/mg and 6.6 units/mg for for PKA and PKG, respectively[1].
A statistically significant effect of isoprenaline on the activity ratio of guinea-pig heart was only: observed with Malantide[1].
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