Chymase-IN-1
CAS No. : 862090-74-2
| Size | Price | Stock |
|---|---|---|
| 1mg | $447 | Get quote |
| 5 mg | Get quote | |
| 10 mg | Get quote | |
| We match the lowest price on market. | ||
We offer a substantial discount on larger orders, please inquire via [email protected]
or Fax: (86)21-58955996
Inquiry for price and availability only. Please place your order via our email or fax.
| Cat. No. : | HY-100269 |
| M.Wt: | 431.83 |
| Formula: | C20H15ClNO4PS |
| Purity: | >98 % |
| Solubility: | 10 mM in DMSO |
Chymase-IN-1 is a potent, selective, orally active, nonpeptide inhibitor of human mast cell chymase with an IC50 of 29 nM. IC50 & Target: IC50: 29 nM (chymase)[1] In Vitro: Chymase-IN-1 (compound 5f) is a potent, selective, orally active, nonpeptide inhibitor of human mast cell chymase with an IC50 of 29 nM. Results demonstrate that Chymase-IN-1 has a chymase Ki value of 36 nM and a Cat G Ki value of 9500 nM[1]. In Vivo: Chymase-IN-1 exhibits low oral bioavailability in rats (F=3%; oral t1/2=1.8 h)[1].
Lorem ipsum dolor sit amet, consectetur adipisicing elit. Autem earum hic iste maiores, nam neque rem suscipit. Adipisci consequatur error exercitationem fugit ipsam optio qui, quibusdam repellendus sed vero! Debitis.
Inquiry Information- Product Name:
- Chymase-IN-1
- Cat. No.:
- HY-100269
- Quantity:
Your information is safe with us.