DG-041
CAS No. : 861238-35-9
| Size | Price | Stock |
|---|---|---|
| 5mg | $125 | In-stock |
| 10mg | $198 | In-stock |
| 25mg | $420 | In-stock |
| 50mg | $670 | In-stock |
| 100mg | $980 | In-stock |
| 200 mg | Get quote | |
| 500 mg | Get quote | |
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| Cat. No. : | HY-10835 |
| M.Wt: | 592.32 |
| Formula: | C23H15Cl4FN2O3S2 |
| Purity: | >98 % |
| Solubility: | DMSO : 250 mg/mL (ultrasonic) |
DG-041 is a potent, high affinity and selective EP3 receptor antagonist with IC50s of 4.6 nM and 8.1 nM in the binding and FLIPR assay, respectively. DG-041 inhibits PGE2 facilitation of platelet aggregation. DG-041 crosses the blood-brain barrier[1][2]. In Vitro: DG-041 was a less potent antagonist of the DP1 (IC50=131 nM), EP1 (IC50=486 nM), and TP receptors (IC50=742 nM)[1]. In Vivo: DG-041 (1.78 mg/kg for intravenous or 9.62 mg/kg for oral) has t1/2 of 2.7 hours, 4.06 hours and Cmax of 9.46 μM, 2.74 μM for intravenous and oral administration, respectively. DG-041 has CL of 1250 mL/h/kg for intravenous[1].
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- DG-041
- Cat. No.:
- HY-10835
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