PU-H39
CAS No. : 852030-38-7
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| Cat. No. : | HY-121723 |
| M.Wt: | 378.28 |
| Formula: | C16H13Cl2N5S |
| Purity: | >98 % |
| Solubility: |
PU-H39 (compound 9g) is a selective Grp94 inhibitor with an IC50 of 0.12 μM. PU-H39 exhibits 34% and 32% inhibition of MKNK2 and ROCK2 kinases respectively at 10 μM. PU-H39 can be used for the research of breast cancer[1].
In Vitro:PU-H39 (compound 9g) (0.12 μM (Grp94), >300 μM (Hsp90α/β), 145.4 μM (Trap-1); 24 h at 4 °C) potently and selectively inhibits Grp94 with an IC50 of 0.12 μM[1].
PU-H39 (compound 9g) (10 μM; 1 h incubation, 30 min elution) shows minimal off-target binding to kinases at 10 μM, with only weak inhibition of MKNK2 and ROCK2 observed[1].
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