ADL5859
CAS No. : 850305-06-5
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| Cat. No. : | HY-14356 |
| M.Wt: | 392.49 |
| Formula: | C24H28N2O3 |
| Purity: | >98 % |
| Solubility: |
ADL-5859 is a selective and orally active δ opioid receptor (DOR) agonist with an Ki and an EC50 value of 0.84 and 20 nM, respectively. ADL-5859 also shows inhibitory activity to hERG channel with an IC50 value of 78 μM. ADL-5859 can be used for the research of pain[1][2]. IC50 & Target:IC50: 78 μM (hERG channel), 43 μM (CYP2D6)[1][2] In Vitro:ADL-5859 (0-10 μM) shows activities to δ opioid receptor with an Ki and an EC50 value of 0.84 and 20 nM, and inhibits 32% and 37% activities to µ and κ opioid receptor, respectively[1]. ADL-5859 (0-100 μM) exhibits inhibitory activity to hERG channel with an IC50 value of 78 μM[1]. ADL-5859 (0-100 μM) inhibits activity of the drug metabolizing enzyme cytochrome P450 2D6 (CYP2D6) in vitro with an IC50 value of 43 μM[2].
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- ADL5859
- Cat. No.:
- HY-14356
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