Enalaprilat (dihydrate)
CAS No. : 84680-54-6
(Synonyms: MK-422)
| Size | Price | Stock |
|---|---|---|
| 50mg | $60 | In-stock |
| 100mg | $105 | In-stock |
| 500mg | $420 | In-stock |
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| Cat. No. : | HY-B0231 |
| M.Wt: | 384.42 |
| Formula: | C18H28N2O7 |
| Purity: | >98 % |
| Solubility: | H2O : 12.5 mg/mL (ultrasonic);DMSO : 100 mg/mL (ultrasonic) |
Enalaprilat dihydrate (MK-422), the active metabolite of the oral prodrug Enalapril, is a potent, competitive and long-acting angiotensin-converting enzyme (ACE) inhibitor, with an IC50 of 1.94 nM. Enalaprilat dihydrate can be used for the research of hypertension[1][2][3]. IC50 & Target: IC50: 1.94 nM (ACE)[1] In Vitro: Enalaprilat (1 nM-10 μM; 24 h) dihydrate attenuates the IGF-I induced neonatal rat cardiac fibroblast growth (30% reduction) in a concentration-dependent fashion, with an IC50 of 90 mM[2]. In Vivo: Enalaprilat (0.01%-2.9% in the eyedrop solution) dihydrate shows significant intraocular pressure (IOP)-lowering effect in rabbits[3].
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