CAY10471 (Racemate)
CAS No. : 844639-57-2
(Synonyms: TM30089 (Racemate))
| Size | Price | Stock |
|---|---|---|
| 5mg | $90 | In-stock |
| 10mg | $140 | In-stock |
| 25mg | $290 | In-stock |
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| Cat. No. : | HY-13706 |
| M.Wt: | 416.47 |
| Formula: | C21H21FN2O4S |
| Purity: | >98 % |
| Solubility: | DMSO : 150 mg/mL (ultrasonic) |
CAY10471 Racemate (TM30089 Racemate) is a potent and highly selective prostaglandin D2 receptor CRTH2 antagonist, with a Ki of 0.6 nM for hCRTH2, selective over human thromboxane A2 receptor TP (Ki, >10000 nM) or PGD2 receptor DP (Ki, 1200 nM). CAY10471 Racemate also has effect on mouse and rat orthologs of CRTH2[1]. IC50 & Target:Ki: 0.6 nM (CRTH2), 1200 nM (DP)[1] In Vitro: CAY10471 Racemate (Compound 13) inhibits PGD2-induced inositol phosphate or cAMP formation, suppresses β-arrestin translocation with IC50s of 12 and 3 nM, respectively[1].
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