Racecadotril
CAS No. : 81110-73-8
(Synonyms: Acetorphan)
| Size | Price | Stock |
|---|---|---|
| 200mg | $66 | In-stock |
| 500mg | $98 | In-stock |
| 1g | $117 | In-stock |
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| 10 g | Get quote | |
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| Cat. No. : | HY-17399 |
| M.Wt: | 385.48 |
| Formula: | C21H23NO4S |
| Purity: | >98 % |
| Solubility: | DMSO : ≥ 100 mg/mL |
Racecadotril (Acetorphan) is a neutral endopeptidase (NEP) inhibitor. Racecadotril and its active metabolite Thiorphan inhibits purified NEP activity from mouse brain with Kis of 4500 and 6.1 nM, , respectively. Antidiarrheal agent[1].
In Vivo: In mice, following i.v. administration, Racecadotril is rapidly metabolized to Thiorphan; thus, 30 min after the injection only Thiorphan is recovered from the kidney whereas the parent compound Racecadotril is not detected[1].
In rats 92% of a single-dose (10 mg/kg) of radioactively labeled Racecadotril is eliminated within 24 h[1].
Racecadotril is a neutral endopeptidase (NEP) inhibitor with known antidiarrheal activity in animals. Orally administered Racecadotril (100 mg/kg ) shows efficacy in a rat model of castor oil-induced diarrhea[2].
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