Cisapride
CAS No. : 81098-60-4
(Synonyms: R 51619; (±)-Cisaprid)
| Size | Price | Stock |
|---|---|---|
| 5mg | $50 | In-stock |
| 10mg | $79 | In-stock |
| 50mg | $125 | In-stock |
| 100mg | $198 | In-stock |
| 200mg | $317 | In-stock |
| 500 mg | Get quote | |
| 1 g | Get quote | |
| We match the lowest price on market. | ||
We offer a substantial discount on larger orders, please inquire via [email protected]
or Fax: (86)21-58955996
Inquiry for price and availability only. Please place your order via our email or fax.
| Cat. No. : | HY-14149 |
| M.Wt: | 465.95 |
| Formula: | C23H29ClFN3O4 |
| Purity: | >98 % |
| Solubility: | H2O : < 0.1 mg/mL;DMSO : 100 mg/mL (ultrasonic) |
Cisapride (R 51619) is an orally active 5-HT4 receptor agonist with an EC50 value of 140 nM. Cisapride is a hERG blocker with an IC50 value of 9.4 nM. Cisapride is a gastroprokinetic agent that stimulates gastrointestinal motor activity[1][2][3][4]. In Vitro:Cisapride (1-100 nM) is a potent hERG blockers with an IC50 value of 9.4 nM[1]. Cisapride (1-100 nM) shows efficacy to 5-HT4 receptor with an EC50 value of 140 nM[1]. Cisapride (0.3, 1, 3, 10 and 30 μM) dose-dependently inhibits Kv4.3 with an IC50 value of 9.8 μM in Kv4.3 potassium channels expressing CHO cells[2]. In Vivo:Cisapride (0.1-1 mg/kg; i.v., once) stimulates antral and colonic motility in conscious dogs[3]. Cisapride (2 mg/kg (i.p.); 4 mg/kg, (oral administration); once) shows no significant differences in macroscopic features, histopathological features, cytokines profile and bodyweight changes with TNBS-treated rats[4].
Lorem ipsum dolor sit amet, consectetur adipisicing elit. Autem earum hic iste maiores, nam neque rem suscipit. Adipisci consequatur error exercitationem fugit ipsam optio qui, quibusdam repellendus sed vero! Debitis.
Inquiry Information- Product Name:
- Cisapride
- Cat. No.:
- HY-14149
- Quantity:
Your information is safe with us.