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|---|---|---|
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| 500 mg | Get quote | |
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| Cat. No. : | HY-121122 |
| M.Wt: | 359.46 |
| Formula: | C23H25N3O |
| Purity: | >98 % |
| Solubility: |
A778317 is a TRPV1 antagonists. A778317 can block changes in intracellular calcium levels mediated by TRPV1 receptors, with a pIC50 value of 8.31. A-778317 can also block the activation of natural rat TRPV1 receptors in dorsal root ganglion neurons by capsaicin and acid[1].
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