Basimglurant (Standard)
CAS No. : 802906-73-6
(Synonyms: RG7090 (Standard); RO4917523 (Standard))
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| Cat. No. : | HY-15446R |
| M.Wt: | 325.77 |
| Formula: | C18H13ClFN3 |
| Purity: | >98 % |
| Solubility: |
Basimglurant (RG7090; RO4917523) (Standard) is the analytical standard of Basimglurant. This product is intended for research and analytical applications. Basimglurant is a selective, orally active, blood-brain barrier permeable negative allosteric modulator of metabotropic glutamate receptor 5 (mGluR5), with a Ki of 1.4 nM (against [3H]-ABP688 (HY-110141)) and 35.6 nM (against [3H]-MPEP (HY-14609A)). Basimglurant inhibits mGlu5-mediated signaling pathways and receptor constitutive activity, regulates dopamine levels in the nucleus accumbens, exerts anxiolytic, antidepressant-like, analgesic and arousal-promoting effects, and alters δ-wave power during non-rapid eye movement sleep. Basimglurant can be used in research on depression, fragile X syndrome, anxiety disorders, etc.[1][2] IC50 & Target:Kd: 1.1 nM (mGlu5)[1]
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