GEMSA
CAS No. : 77482-44-1
(Synonyms: 2-Guanidinoethylmercaptosuccinic acid)
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| Cat. No. : | HY-118120 |
| M.Wt: | 235.26 |
| Formula: | C7H13N3O4S |
| Purity: | >98 % |
| Solubility: | 10 mM in DMSO |
GEMSA (2-Guanidinoethylmercaptosuccinic acid) is a potent specific inhibitor of carboxypeptidase B-like processing enzyme (encephalin convertase) with the Ki value of 8.8 nM[1][2][3]. IC50 & Target: Encephalin convertase, Ki 值为8.8 nM. In Vitro: GEMSA inhibits the activation of TAFI and porcine CBB[1]. GEMSA can inhibit the prolongation of lysis time in recombinant BAP and does not lead to the lysis of APC fibronectin[1]. GEMSA inhibits the prolongation of lysis time in porcine CPB, TAFI, and recombinant BAP, APC with the EC50 values of 0.34 μM, 100μM, 115 μM, 90 μM respectively[1][2]. In Vivo: GEMSA (ICV, 0.1μg/mg, every, 3days) results in a 75% increase in hypothalamic luteinizing hormone-releasing hormone and serum luteinizing hormone levels, and a 60% decrease in serum prolactin concentrations in rat[3]
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