ORM-10962
CAS No. : 763926-98-3
| Size | Price | Stock |
|---|---|---|
| 5mg | $600 | In-stock |
| 10mg | $1000 | In-stock |
| 50mg | $3500 | In-stock |
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| Cat. No. : | HY-123785 |
| M.Wt: | 459.54 |
| Formula: | C27H29N3O4 |
| Purity: | >98 % |
| Solubility: | DMSO : 250 mg/mL (ultrasonic) |
ORM-10962 is a potent, highly selective sodium-calcium exchanger (NCX) inhibitor, with IC50 values of 67 and 55 nM for the reverse and forward mode inhibition, respectively. ORM-10962 shows antiarrhythmic effect[1][2][3]. IC50 & Target: NCX[1][2]. In Vitro: ORM-10962 (10 nM, 100 nM and 1 μM) decreased the NCX current in dog ventricular myocytes in a concentration-dependent manner with estimated IC50 values of 55 and 67 nM at -80 and at 20 mV, respectively[1]. In Vivo: ORM-10962 (0.3 mg/kg, IV, once) pre-treatment significantly delays the development and recurrence of ventricular extrasystoles (by about 50%) or ventricular tachycardia (by about 30%) in anesthetized guinea pigs[1].
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