Antitrypanosomal agent 1
CAS No. : 75144-12-6
| Size | Price | Stock |
|---|---|---|
| 1g | $50 | In-stock |
| 5g | $133 | In-stock |
| 10g | $266 | In-stock |
| 50 g | Get quote | |
| 100 g | Get quote | |
| We match the lowest price on market. | ||
We offer a substantial discount on larger orders, please inquire via [email protected]
or Fax: (86)21-58955996
Inquiry for price and availability only. Please place your order via our email or fax.
| Cat. No. : | HY-W052512 |
| M.Wt: | 282.60 |
| Formula: | C11H14Cl3NO |
| Purity: | >98 % |
| Solubility: | H2O : 10 mg/mL (ultrasonic);DMSO : 25 mg/mL (ultrasonic) |
Antitrypanosomal agent 1 is a potent and selective trypanothione reductase (TR) inhibitor with an IC50 of 3.3 μM. Antitrypanosomal agent 1 inhibits glutathione reductase (GR) (IC50=64.8 μM) and T. brucei (EC50=1 μM). Antitrypanosomal agent 1 has anti-trypanosomal activity[1].
IC50 & Target: IC50: 3.3 μM (trypanothione reductase) and 64.8 μM (glutathione reductase)[1]
EC50: 1 μM (T. brucei)[1]
In Vitro: Antitrypanosomal agent 1 (compound 8a) has an selectivity for TR (GR IC50/TR IC50) of 20[1].
Lorem ipsum dolor sit amet, consectetur adipisicing elit. Autem earum hic iste maiores, nam neque rem suscipit. Adipisci consequatur error exercitationem fugit ipsam optio qui, quibusdam repellendus sed vero! Debitis.
Inquiry Information- Product Name:
- Antitrypanosomal agent 1
- Cat. No.:
- HY-W052512
- Quantity:
Your information is safe with us.