Bepridil (hydrochloride hydrate)
CAS No. : 74764-40-2
(Synonyms: (±)-Bepridil (hydrochloride hydrate); Org 5730 (hydrochloride hydrate))
| Size | Price | Stock |
|---|---|---|
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| 5mg | $60 | In-stock |
| 10mg | $100 | In-stock |
| 25mg | $220 | In-stock |
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| Cat. No. : | HY-16952A |
| M.Wt: | 421.02 |
| Formula: | C24H37ClN2O2 |
| Purity: | >98 % |
| Solubility: | DMSO : 125 mg/mL (ultrasonic) |
Bepridil hydrochloride hydrate ((±)-Bepridil hydrochloride hydrate) is a non-selective, long-acting Ca+ channel antagonist and Na+, K+ channel inhibitor, with antianginal and type I antiarrhythmic effects. Bepridil hydrochloride hydrate also acts as a cardiac Na+/Ca2+ exchange (NCX1) inhibitor. Bepridil hydrochloride hydrate can be used for the research of cardiovascular disorders[1][2][3][4][5].
In Vitro: Bepridil hydrochloride hydrate blockades of Ca2+-dependent action potentials in vascular smooth muscle of dog coronary artery[2].
Bepridil hydrochloride hydrate blocks Ca currents and Na currents with IC50s of 0.5 μM and 30 μM, respectively in cultured ventricular cells[4].
Bepridil hydrochloride hydrate decreases IKs under blockade of IKr with E4031 (5 μM), in a concentration-dependent manner[5].
In Vivo: Bepridil hydrochloride hydrate exhibits a half-life of averages 33±15 hours after single-dose administration[6].
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