SKF-82958 (hydrobromide)
CAS No. : 74115-01-8
(Synonyms: (±)-SKF-82958 (hydrobromide); Chloro-APB (hydrobromide))
| Size | Price | Stock |
|---|---|---|
| 5mg | $119 | In-stock |
| 10mg | $192 | In-stock |
| 25mg | $384 | In-stock |
| 50mg | $696 | In-stock |
| 100mg | $1260 | In-stock |
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| Cat. No. : | HY-10435A |
| M.Wt: | 410.73 |
| Formula: | C19H21BrClNO2 |
| Purity: | >98 % |
| Solubility: | DMSO : ≥ 100 mg/mL |
SKF-82958 ((±)-SKF 82958) hydrobromide is a dopamine D1 receptor full agonist (K0.5=4 nM), displays selective for D1 over D2 receptors (K0.5=73 nM). SKF-82958 hydrobromide induces dopamine D1 receptor-dependent adenylate cyclase activity in rat striatal membranes (EC50=491 nM)[1].
In Vivo: SKF-82958 ((±)-SKF 82958) hydrobromide (0.003-0.1 mg/kg; i.p.) results in dose-dependent increases in responding on the SKF-82958 appropriate lever, with full substitution following administration of the SKF-82958 hydrobromide training dose 0.03 mg/kg. Increasing the dose of SKF-82958 hydrobromide also results in a significant reduction in response rate[2].
SKF-82958 hydrobromide (0.5-2.0 mg/kg; i.p) significantly suppresses pilocarpine-induced jaw movements[3].
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