Fenoldopam (mesylate)
CAS No. : 67227-57-0
(Synonyms: Fenoldopam (methanesulfonate); SKF-82526 (mesylate))
| Size | Price | Stock |
|---|---|---|
| 5mg | $35 | In-stock |
| 10mg | $55 | In-stock |
| 25mg | $116 | In-stock |
| 50mg | $187 | In-stock |
| 100mg | $286 | In-stock |
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| Cat. No. : | HY-B0735A |
| M.Wt: | 401.86 |
| Formula: | C17H20ClNO6S |
| Purity: | >98 % |
| Solubility: | H2O : 10 mg/mL (ultrasonic);DMSO : ≥ 36 mg/mL |
Fenoldopam mesylate (SKF-82526) is a D1 receptor agonist and a novel lysine-specific demethylase 1 (LSD1) inhibitor (IC50=0.8974 μM). Fenoldopam mesylate shows anti-hypertensive effects, anti-cancer cell proliferation activity and can induce cells apoptosis[1][2][3].
IC50 & Target:IC50: 0.8974 μM (LSD1)[2]
In Vitro: Fenoldopam is a partial agonist with low efficacy at DA1 receptors linked to cAMP generation in the LLC-PK1 cells[1].
Fenoldopam (0-300 μM; 48 or 72 h) displays significant antiproliferative activity against RCC cell lines[2].
Fenoldopam (5 μM and 10 μM; 72 h) induces cell apoptosis in a dose-dependent manner[2].
In Vivo: Fenoldopam mesylate (subcutaneous injection; 100 mg/kg; once daily; 2 d) can induce arteritis in rats detected by magnetic resonance imaging (MRI)[3].
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