Cloxacepride
CAS No. : 65569-29-1
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| Cat. No. : | HY-106645 |
| M.Wt: | 468.37 |
| Formula: | C22H27Cl2N3O4 |
| Purity: | >98 % |
| Solubility: | 10 mM in DMSO |
Cloxacepride is an orally active and potent antiallergic agent. Cloxacepride is a CaM (calmodulin) antagonist. Cloxacepride has anti-PCA (passive cutaneous anaphylaxis) activity[1][2].
In Vitro:Cloxacepride (10-50 μM) shows inhibitory effect on Compound 48/80 (HY-115768)-induced histamine and serotonin release from rat mesenterial mast cells. The IC50 is determined to 21 μM (histamine) and 19 μM (serotonin)[3].
In Vivo:Oral ED50 values for cloxacepride of 46-49 mg/kg were comparable to that of theophylline (HY-B0809) and to an intravenous injection of 2 mg/kg of disodium chromoglycate (DSCG) followed by immediate challenge[1].
Cloxacepride has anti-PCA activity when administered orally 15 or 60 min before antigenic challenge[1].
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