Mosapride (citrate dihydrate)
CAS No. : 636582-62-2
(Synonyms: TAK-370 (citrate dihydrate); AS-4370 (citrate dihydrate))
| Size | Price | Stock |
|---|---|---|
| 5mg | $30 | In-stock |
| 10mg | $44 | In-stock |
| 25mg | $75 | In-stock |
| 50mg | $120 | In-stock |
| 100mg | $180 | In-stock |
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| Cat. No. : | HY-B0189B |
| M.Wt: | 650.05 |
| Formula: | C27H37ClFN3O12 |
| Purity: | >98 % |
| Solubility: | 10 mM in DMSO |
Mosapride (TAK-370) citrate dehydrate is a gastroprokinetic agent with 5-hydroxytryptamine4 receptor agonist activity and has been widely used in the research of a variety of gastrointestinal disorders. Mosapride citrate dihydrate potently inhibits Kv4.3 in a concentration-dependent manner with IC50 values of 15.2 μM[1]. Mosapride citrate dihydrateselectively stimulates upper GI motility in vivo[2]. IC50 & Target:IC50: 15.2 μM Kv4.3[1] In Vitro: Mosapride (0.3-30 μM) exhibits an inhibitory activity against Kv4.3 with an IC50 of 15.2 μM in a concentration-dependent manner. Mosapride also inhibits the open state of Kv4.3 currents during depolarization and accelerates the closed-state inactivation at subthreshold potentials[1]. In Vivo: Mosapride (Intravenous injection;0.3-3 mg/kg) dose-dependently increases the antral motor activity in conscious dogs which indicates that mosapride selectively stimulates upper gastrointestinal motility[2].
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