| Size | Price | Stock |
|---|---|---|
| 5mg | $145 | In-stock |
| 10 mg | Get quote | |
| 50 mg | Get quote | |
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| Cat. No. : | HY-100704 |
| M.Wt: | 326.82 |
| Formula: | C16H23ClN2O3 |
| Purity: | >98 % |
| Solubility: | 10 mM in DMSO |
Procaterol hydrochloride is a selective intermediate-acting β2 adrenoreceptor agonist with an EC50 of 12.9 µM[1]. Procaterol hydrochloride can inhibit inflammation both in vivo and in vitro[2].
In Vitro: Procaterol treat inflammation through inhibiting oxidative stress in vitro[2].
Procaterol (25-200 nM) increases the viability of 16HBE cells[2].
In Vivo: Procaterol significantly increases conditioned stimulus (CS)-evoked freezing levels[3]. Propranolol-mediated blockade of β-adrenergic receptors (β-ARs) significantly reduces behavioral expression of Pavlovian threat conditioning (PTC), whereas systemic activation of β2-ARs using Procaterol enhances it[3].
Procaterol hydrochloride is freshly dissolved in 0.9% sterile saline immediately prior to injections[3].
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