Dibucaine (hydrochloride)
CAS No. : 61-12-1
(Synonyms: Cinchocaine hydrochloride)
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| Cat. No. : | HY-B0552A |
| M.Wt: | 379.92 |
| Formula: | C20H30ClN3O2 |
| Purity: | >98 % |
| Solubility: | DMSO : 110 mg/mL (ultrasonic);H2O : 100 mg/mL (ultrasonic) |
Dibucaine hydrochloride (Cinchocaine hydrochloride) is a sodium channel inhibitor. Dibucaine hydrochloride is a potent SChE inhibitor[1][2]. In Vitro: Dibucaine hydrochloride (Cinchocaine hydrochloride) reduced the degradation of BSA-gold complex in the reservosomes, which was not caused either by an inhibition of the whole proteolytic activity of the parasite or by a reduction on the expression levels of cruzipain[1]. Dibucaine, a quaternary ammonium compound, inhibited SChE to a minimum within 2 min in a reversible manner. The inhibition was very potent. It had an IC(50) of 5.3 microM with BuTch or 3.8 microM with AcTch. The inhibition was competitive with respect to BuTch with a K(i) of 1.3 microM and a linear-mixed type (competitive/noncompetitive) with respect to AcTch with inhibition constants, K(i) and K(I) of 0.66 and 2.5 microM, respectively. Dibucaine possesses a butoxy side chain that is similar to the butryl group of BuTch and longer by an ethylene group from AcTch[2].
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