Tasimelteon
CAS No. : 609799-22-6
(Synonyms: BMS-214778; VEC-162)
| Size | Price | Stock |
|---|---|---|
| 5mg | $30 | In-stock |
| 10mg | $48 | In-stock |
| 25mg | $84 | In-stock |
| 50mg | $140 | In-stock |
| 100mg | $230 | In-stock |
| 500mg | $565 | In-stock |
| 1 g | Get quote | |
| 5 g | Get quote | |
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| Cat. No. : | HY-14803 |
| M.Wt: | 245.32 |
| Formula: | C15H19NO2 |
| Purity: | >98 % |
| Solubility: | DMSO : ≥ 33 mg/mL |
Tasimelteon (BMS-214778) is an orally active and selective dual melatonin receptor agonist (DMRA). Tasimelteon has 2.1-4.4 times greater affinity for the MT2 receptor than for the MT1 receptor. Tasimelteon is a circadian regulator and has the potential for Non-24-Hour Sleep-Wake Disorder (Non-24)[1][2]. In Vitro: Tasimelteon (BMS-214778) has 2.1-4.4 times greater affinity for the MT2 receptor believed to mediate circadian rhythm phase-shifting (Ki=0.0692 nM and Ki=0.17 nM in NIH-3T3 and CHO-K1 cells, respectively), than for the MT1 receptor (Ki=0.304 nM and Ki=0.35 nM, respectively). Tasimelteon has no appreciable affinity for more than 160 other pharmacologically relevant receptors and several enzymes[1].
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