| Size | Price | Stock |
|---|---|---|
| 5g | $29 | In-stock |
| 10g | $57 | In-stock |
| 25g | $112 | In-stock |
| 100g | $446 | In-stock |
| 200 g | Get quote | |
| 500 g | Get quote | |
| We match the lowest price on market. | ||
We offer a substantial discount on larger orders, please inquire via [email protected]
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| Cat. No. : | HY-W015239 |
| M.Wt: | 189.17 |
| Formula: | C10H7NO3 |
| Purity: | >98 % |
| Solubility: | DMSO : 100 mg/mL (ultrasonic) |
KAT8-IN-1 is a lysine (K) acetyltransferase 8 (KAT8) inhibitor, with IC50s of 141 μM (KAT8), 221 μM (KAT2B), 106 μM (KAT3B), respectively. KAT8 inhibits histone acetyltransferases (HATs), and could result in disease states, such as cancer or inflammatory diseases[1].
IC50 & Target: IC50: 141 μM (KAT8), 221 μM (KAT2B), 106 μM (KAT3B)[1]
In Vitro: KAT8-IN-1 (compound 19) losses anti-oxidant activity (EC50>1 mM)[1].
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