Clebopride (malate)
CAS No. : 57645-91-7
| Size | Price | Stock |
|---|---|---|
| 5mg | $60 | In-stock |
| 10mg | $84 | In-stock |
| 25mg | $135 | In-stock |
| 50mg | $180 | In-stock |
| 100mg | $300 | In-stock |
| 200 mg | Get quote | |
| 500 mg | Get quote | |
| We match the lowest price on market. | ||
We offer a substantial discount on larger orders, please inquire via [email protected]
or Fax: (86)21-58955996
Inquiry for price and availability only. Please place your order via our email or fax.
| Cat. No. : | HY-B1613A |
| M.Wt: | 507.96 |
| Formula: | C24H30ClN3O7 |
| Purity: | >98 % |
| Solubility: | H2O : 8.33 mg/mL (ultrasonic);DMSO : 60 mg/mL (ultrasonic) |
Clebopride malate is an orally active dopamine Receptor antagonist. Clebopride malate acts on dopamine D2 receptors and has antiemetic and prokinetic effects. Clebopride malate can be used in the study of functional gastrointestinal disorders[1][2][3].
In Vitro:Clebopride malate (0.1 nM-10μM, 30 min) selectively binds to D2 dopamine receptors (Ki: 3.5 nM) and α2 adrenergic receptors (Ki: 780 nM) in bovine brain membranes[3].
Clebopride malate inhibits ETS-induced gastric strip contractions (IC50: 0.43 μM) [3].
Lorem ipsum dolor sit amet, consectetur adipisicing elit. Autem earum hic iste maiores, nam neque rem suscipit. Adipisci consequatur error exercitationem fugit ipsam optio qui, quibusdam repellendus sed vero! Debitis.
Inquiry Information- Product Name:
- Clebopride (malate)
- Cat. No.:
- HY-B1613A
- Quantity:
Your information is safe with us.