TD-5471
CAS No. : 530084-87-8
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| Cat. No. : | HY-19942 |
| M.Wt: | 521.61 |
| Formula: | C32H31N3O4 |
| Purity: | >98 % |
| Solubility: |
TD-5471 is a potent and selective full agonist of the human β2-adrenoceptor[1]. IC50 & Target:β2 adrenoceptor[1] In Vitro:TD-5471 is potent, with slow onset in an in vitro guinea pig trachea model. TD-5471 has potency with pEC50 of 8.7 in the guinea pig tracheal ring assay.TD-5471 is structurally differentiated from Milveterol (HY-14297) and its long duration of action is consistent with a correlation with hydrophobicity observed in other long-acting β2-agonist discovery programs[1]. In Vivo:TD-5471 shows a dose-dependent and long duration of action in an in vivo guinea pig model of bronchoprotection. In a guinea pig model of in vivo bronchoprotection, TD-5471 shows excellent potency (measured 1.5 h after nebulized dosing). TD-5471-mediated bronchoprotection at 72 h is dose-dependent[1].
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- Cat. No.:
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