NS5806
CAS No. : 426834-69-7
| Size | Price | Stock |
|---|---|---|
| 1mg | $50 | In-stock |
| 5mg | $120 | In-stock |
| 10mg | $190 | In-stock |
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| 100 mg | Get quote | |
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| Cat. No. : | HY-108588 |
| M.Wt: | 574.07 |
| Formula: | C16H8Br2F6N6O |
| Purity: | >98 % |
| Solubility: | DMSO : 250 mg/mL (ultrasonic) |
NS5806, a potent potassium current activator, increases KV4.3/KChIP2 peak current amplitudes with an EC50 of 5.3 μM. NS5806 slows KV4.3 and KV4.2 current dacay in channel complexes containing KChIP2[1].
IC50 & Target: IC50: 5.3 nM (KV4.3)[1]
In Vitro: NS5806 (10 µM) induces a 65% increase of KV4.3/KChIP2/DPP6 peak current amplitudes concentration-dependently and the time course of inactivation (τ) is slowed with an EC50 value of 25.4 µM in CHO-K1 cells[1].
NS5806 activates canine transient outward potassium current (Ito) with an IC50 of 40.7 nM and an EC50 of 1.6 nM for inhibition and stimulation on rabbit, respectively[2].
NS5806 (10-100 nM) has concentration-dependent effects on ventricular and atrial Ito[2].
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