H2L 5765834
CAS No. : 420841-84-5
| Size | Price | Stock |
|---|---|---|
| 1mg | $71 | In-stock |
| 5mg | $150 | In-stock |
| 10mg | $240 | In-stock |
| 25mg | $450 | In-stock |
| 50mg | $670 | In-stock |
| 100mg | $950 | In-stock |
| 200 mg | Get quote | |
| 500 mg | Get quote | |
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| Cat. No. : | HY-15706 |
| M.Wt: | 404.33 |
| Formula: | C21H12N2O7 |
| Purity: | >98 % |
| Solubility: | DMSO : 250 mg/mL (ultrasonic) |
H2L 5765834 is an antagonist of lysophosphatidic acid receptors LPA1, LPA3, and LPA5, with IC50s of 94, 752, and 463 nM respectively[1].
IC50 & Target: IC50: 94 nM (LPA1), 752 nM (LPA3), and 463 nM (LPA5)[1]
In Vitro: H2L 5765834 displays no effect on LPA2 or LPA4 receptors[1].
H2L 5765834 inhibits LPA-induced platelet shape change with an IC50 of 13.73±2.52 μM[1].
In Vivo: H2L 5765834 (20 mg/kg; i.p.) could not affect the LPA-induced decrease of alanine transaminase (ALT) in the acetaminophen (APAP) overdose-induced acute liver injury model[2].
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