Grapiprant
CAS No. : 415903-37-6
(Synonyms: CJ-023423; RQ-00000007; AAT-007)
| Size | Price | Stock |
|---|---|---|
| 5mg | $90 | In-stock |
| 10mg | $150 | In-stock |
| 25mg | $250 | In-stock |
| 50mg | $450 | In-stock |
| 100mg | $720 | In-stock |
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| Cat. No. : | HY-16781 |
| M.Wt: | 491.61 |
| Formula: | C26H29N5O3S |
| Purity: | >98 % |
| Solubility: | DMSO : ≥ 50 mg/mL |
Grapiprant (CJ-023423) is a selective EP4 receptor antagonist whose physiological ligand is prostaglandin E2 (PGE2). Grapiprant displaces [3H]-PGE2 (1 nM) binding to dog recombinant EP4 receptor with IC50 value of 35 nM and Ki value of 24 nM. Grapiprant has the potential for osteoarthritic pain and inflammation treatment[1][2][3] . In Vivo: Grapiprant (0-50 mg/kg; oral administration; every 24 hours; for 9 months; beagles) is safe for dogs by long-term oral administration. Efficacy of Grapiprant in the treatment of dogs with osteoarthritis needs to be evaluated in other studies[3] .
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