NP118809
CAS No. : 41332-24-5
(Synonyms: 39-1B4)
| Size | Price | Stock |
|---|---|---|
| 100mg | $96 | In-stock |
| 200mg | $120 | In-stock |
| 500mg | $150 | In-stock |
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| 5 g | Get quote | |
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| Cat. No. : | HY-14462 |
| M.Wt: | 460.61 |
| Formula: | C32H32N2O |
| Purity: | >98 % |
| Solubility: | DMSO : 50 mg/mL (ultrasonic) |
NP118809 is a potent N-type calcium channel blocker, with an IC50 of 0.11 μM; also less potently inhibits L-type calcium channel with an IC50 of 12.2 μM. IC50 & Target: IC50: 0.11 μM (N-type calcium channel), 12.2 μM (L-type calcium channel)[1][2] In Vitro: NP118809 is a potent N-type calcium channel blocker, with an IC50 of 0.11 μM; also inhibits L-type calcium channel with an IC50 of 12.2 μM. NP118809 inhibits the hERG potassium channel in HEK cells, with an IC50 of 7.4 μM[1]. In Vivo: NP118809 (25 mg/kg, i.p.) shows significant analgesic activity in the phase IIA portions of the rat formalin model[1]. NP118809 (30 mg/kg, p.o.) results in 80.3% inhibition of mechanical allodynia and 96.3% inhibition of thermal hyperalgesia in the rat spinal nerve ligation model[2].
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