LPA2 antagonist 2
CAS No. : 36840-10-5
| Size | Price | Stock |
|---|---|---|
| 5mg | $290 | In-stock |
| 10mg | $460 | In-stock |
| 25mg | $750 | In-stock |
| 50mg | $1060 | In-stock |
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| Cat. No. : | HY-113973 |
| M.Wt: | 380.35 |
| Formula: | C20H16N2O6 |
| Purity: | >98 % |
| Solubility: | DMSO : 83.33 mg/mL (ultrasonic) |
LPA2 antagonist 2 (H2L 5226501) is a selective LPA2 antagonist with an IC50 of 28.3 nM and a Ki of 21.1 nM. LPA2 antagonist 2 is >480-fold more selective than LPA3 (IC50 of 13.85 μM)[1]. IC50 & Target: IC50: 28.3 nM (LPA2); 13.85 μM (LPA3)[1] In Vitro: Lysophosphatidic acid (LPA) is a phospholipid mediator that elicits a host of biological effects including cell proliferation, survival, motility and differentiation. LPA has been shown to regulate cancer cell invasion, metastasis, and resistance to both chemotherapeutics and radiation. LPA2 antagonist 2 (H2L 5226501) inhibits LPA1 with an Imax of 59.0% at 30 µM[1].
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