Tolperisone (hydrochloride)
CAS No. : 3644-61-9
| Size | Price | Stock |
|---|---|---|
| 5mg | $32 | In-stock |
| 10mg | $50 | In-stock |
| 50mg | $70 | In-stock |
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| Cat. No. : | HY-B1139 |
| M.Wt: | 281.82 |
| Formula: | C16H24ClNO |
| Purity: | >98 % |
| Solubility: | DMSO : 100 mg/mL (ultrasonic;warming;heat to 60°C);H2O : 100 mg/mL (ultrasonic) |
Tolperisone hydrochloride is a centrally acting muscle relaxant studied in neurological disorders causing pathological rhabdomyosclerosis (pyramidal tract injury, multiple sclerosis, myelopathy, encephalomyelitis), spastic paralysis, and other muscle dystonia-related Encephalopathy. Tolperisone hydrochloride also has antiviral activity[1].
In Vitro:Tolperisone (0-128 μM, 48 h) hydrochloride induces UPR-mediated cancer cell death by directly targeting LSD1, with IC50s of 10-40 μM[1].
Tolperisone inhibits LSD1 activity with an IC50 of 31.09 µM[1].
Tolperisone (100 μM, 48 h) induces cancer cell cycle arrest and apoptosis in AGS, A375, 8505C, and RKO cells[1].
Tolperisone (100 μM, 12 h) repolarizes M2 macrophages into M1 phenotype[1].
In Vivo:Tolperisone (25-100 mg/kg) shows antinociceptive effect in partial sciatic nerve ligation (pSNL) evoked neuropathic pain rats[2].
Tolperisone (60 mg/kg, once a day for 1 week) hydrochloride inhibits tumor growth in A375 cell-derived xenograft mouse model[1].
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