Roluperidone
CAS No. : 359625-79-9
(Synonyms: CYR-101; MIN-101; MT-210)
| Size | Price | Stock |
|---|---|---|
| 5mg | $59 | In-stock |
| 10mg | $97 | In-stock |
| 25mg | $195 | In-stock |
| 50mg | $312 | In-stock |
| 100mg | $500 | In-stock |
| 200 mg | Get quote | |
| 500 mg | Get quote | |
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| Cat. No. : | HY-19469 |
| M.Wt: | 366.43 |
| Formula: | C22H23FN2O2 |
| Purity: | >98 % |
| Solubility: | DMSO : 33.33 mg/mL (ultrasonic) |
Roluperidone (CYR-101) is a novel cyclic amide derivative that has high equipotent affinities for 5-HT2A and sigma-2 receptors (Ki of 7.53 nM and 8.19 nM for 5-HT2A and sigma-2, respectively). IC50 & Target: Ki: 7.53 nM (5-HT2A), 8.19 nM (sigma-2)[1] In Vitro: Roluperidone (CYR-101) also shows binding affinity for α1-adrenergic receptors but low or no affinity for muscarinic, cholinergic, and histaminergic receptors. Although Roluperidone (CYR-101) has no affinities for pre- or postsynaptic dopaminergic receptors, it is probable that sigma-2 receptors are implicated in the modulation of dopamine and glutamatergic pathways, as well as in calcium neuronal modulation[1].
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